SCHEMBL28937129

SCHEMBL28937129

COC(=O)c1cccc(NC(=O)c2ccc(Cl)cc2F)n1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1F P30939 2/20 0.62
SORT1 Q99523 2/20 0.52
MAPT P10636 2/20 0.50
CYP11B2 P19099 1/20 0.50
IDH1 O75874 1/20 0.47
ALDH1A1 P00352 2/20 0.47
GRM5 P41594 1/20 0.46
RXFP1 Q9HBX9 2/20 0.46
NPC1 O15118 3/20 0.46
MRGPRX4 Q96LA9 2/20 0.46
RAB9A P51151 3/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
KMT2A Q03164 2/20 0.45
LMNA P02545 1/20 0.45
GAA P10253 1/20 0.45
TP53 P04637 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28937124 0.88 HTR1F (0.61) HTR1FMAPTALDH1A1GRM5RXFP1
SCHEMBL28937119 0.86 HTR1F (0.63) HTR1FSORT1MAPTCYP11B2ALDH1A1
SCHEMBL28808136 0.81 HTR1F (0.57) HTR1FSORT1MAPTCYP11B2ALDH1A1
SCHEMBL28937139 0.80 RXFP1 (0.71) HTR1FMAPTALDH1A1GRM5RXFP1
SCHEMBL935048 0.79 GRM5 (0.52) IDH1ALDH1A1GRM5NPC1MRGPRX4
SCHEMBL28937138 0.78 HTR1F (0.58) HTR1FMAPTIDH1ALDH1A1GRM5
SCHEMBL21771022 0.77 HTR1F (1.00) HTR1FSORT1CYP11B2NPC1RAB9A
SCHEMBL16317363 0.77 F10 (0.57) CYP11B2ALDH1A1RXFP1NPC1RAB9A
SCHEMBL23702725 0.77 HTR1F (0.60) HTR1FMAPTALDH1A1GRM5NPC1
SCHEMBL23528936 0.77 HTR1F (0.75) HTR1FSORT1CYP11B2ALDH1A1RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110272425-B Pyridyloxyl octahydropyrrolo [3,4-c ] pyrrole derivatives and uses thereof 广东东阳光药业有限公司 2022-11-04 CN disclosed