SCHEMBL28940331

SCHEMBL28940331

CCOC(=O)CCC(Cc1cn(CC)nn1)c1cccc2c1CCN(C(=O)c1ccc(OC)cc1)C2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.37
MAPT P10636 3/20 0.37
HPGD P15428 1/20 0.37
KMT2A Q03164 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
PRMT5 O14744 3/20 0.36
WDR77 Q9BQA1 3/20 0.36
NAMPT P43490 2/20 0.36
STS P08842 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
POLB P06746 1/20 0.35
CDK4 P11802 1/20 0.35
CCND1 P24385 1/20 0.35
CXCR3 P49682 1/20 0.35
KDM4E B2RXH2 1/20 0.34
GLA P06280 1/20 0.34
HTT P42858 1/20 0.34
RAB9A P51151 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
ITGB2 P05107 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28940449 0.90 KEAP1 (0.39) LMNAMAPTHPGDKMT2AHDAC6
SCHEMBL29644375 0.84 KEAP1 (0.45) LMNAMAPTHPGDKMT2AHDAC6
SCHEMBL28739089 0.84 KEAP1 (0.45) LMNAMAPTHPGDKMT2AHDAC6
SCHEMBL28739147 0.82 LMNA (0.37) LMNAMAPTHPGDKMT2AHDAC6
SCHEMBL29644367 0.75 FFAR1 (0.40) LMNAMAPTHPGDKMT2AHDAC6
SCHEMBL28739101 0.75 FFAR1 (0.40) LMNAMAPTHPGDKMT2AHDAC6
SCHEMBL28739006 0.75 KMT2A (0.45) LMNAMAPTHPGDKMT2AHDAC6
SCHEMBL29644435 0.75 KMT2A (0.45) LMNAMAPTHPGDKMT2AHDAC6
SCHEMBL28739042 0.74 NQO1 (0.46) KMT2AGLAALDH1A1
SCHEMBL29644414 0.74 NQO1 (0.46) KMT2AGLAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114507181-A Propionic acid compound containing 5-substituted tetrahydroisoquinoline, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2022-05-17 CN disclosed