SCHEMBL29644367

SCHEMBL29644367

COc1ccc(C(=O)N2CCc3c(cccc3C(CCc3cn(C)nn3)CC(=O)O)C2)cc1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.40
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
KMT2A Q03164 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
PRMT5 O14744 3/20 0.38
WDR77 Q9BQA1 3/20 0.38
KEAP1 Q14145 4/20 0.38
NFE2L2 Q16236 4/20 0.38
NAMPT P43490 1/20 0.37
DRD4 P21917 1/20 0.37
CDK4 P11802 1/20 0.37
CCND1 P24385 1/20 0.37
CXCR3 P49682 1/20 0.36
KCNK3 O14649 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28739101 1.00 FFAR1 (0.40) FFAR1LMNAMAPTHPGDKMT2A
SCHEMBL29644375 0.91 KEAP1 (0.45) FFAR1LMNAMAPTHPGDKMT2A
SCHEMBL28739089 0.91 KEAP1 (0.45) FFAR1LMNAMAPTHPGDKMT2A
SCHEMBL28739147 0.91 LMNA (0.37) LMNAMAPTHPGDKMT2AHDAC6
SCHEMBL28940449 0.83 KEAP1 (0.39) LMNAMAPTHPGDKMT2AHDAC6
SCHEMBL28739082 0.78 FFAR1 (0.51) FFAR1LMNAMAPTHPGDKMT2A
SCHEMBL29644457 0.78 FFAR1 (0.51) FFAR1LMNAMAPTHPGDKMT2A
SCHEMBL28739159 0.78 FFAR1 (0.50) FFAR1LMNAMAPTHPGDKMT2A
SCHEMBL29644336 0.78 FFAR1 (0.50) FFAR1LMNAMAPTHPGDKMT2A
SCHEMBL29201185 0.75 NQO1 (0.55) KEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114507181-B Propionic acid compound containing 5-substituted tetrahydroisoquinoline, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2024-03-26 CN disclosed
CN-114507181-A Propionic acid compound containing 5-substituted tetrahydroisoquinoline, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2022-05-17 CN disclosed