SCHEMBL28940985

SCHEMBL28940985

C[C@@H](O)CNC(=O)c1ccc(OC(N)=O)cn1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 3/20 0.44
CYP2C9 P11712 1/20 0.41
CFTR P13569 1/20 0.41
HPGD P15428 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MAOB P27338 1/20 0.39
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
PARP1 P09874 1/20 0.38
SMPD1 P17405 1/20 0.37
ACVR1 Q04771 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28292586 1.00 SCN9A (0.44) SCN9ACYP2C9CFTRHPGDNPC1
SCHEMBL28941110 0.82 CFTR (0.38) SCN9ACYP2C9CFTRHPGDADORA2A
SCHEMBL28940917 0.82 CFTR (0.38) SCN9ACYP2C9CFTRHPGDADORA2A
SCHEMBL28292566 0.81 MAOB (0.49) SCN9AMAOB
SCHEMBL28963812 0.81 SCN9A (0.40) SCN9ACYP2C9CFTRHPGDNPC1
SCHEMBL28940983 0.81 SCN9A (0.40) SCN9ACYP2C9CFTRHPGDNPC1
SCHEMBL28292577 0.80 CCNC (0.48) SCN9ACYP2C9CFTRHPGDMAOB
SCHEMBL20929477 0.79 ADORA2A (0.44) SCN9AMAOBADORA2AADORA1PARP1
SCHEMBL28284688 0.79 CCNC (0.43) CYP2C9HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL28294317 0.78 SCN9A (0.45) SCN9AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN claimed
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed