SCHEMBL28292566

SCHEMBL28292566

NC(=O)Oc1ccc(C(=O)NCCO)nc1

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.49
MMP13 P45452 1/20 0.41
HIF1A Q16665 5/20 0.41
SCN9A Q15858 1/20 0.40
CNR1 P21554 1/20 0.40
PDE10A Q9Y233 1/20 0.40
MAPT P10636 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28294317 0.85 SCN9A (0.45) MAOBHIF1ASCN9A
SCHEMBL12923703 0.82 PDE10A (0.53) MAOBMMP13HIF1APDE10AL3MBTL1
SCHEMBL28940971 0.82 MMP13 (0.37) MAOBMMP13CNR1MAPTL3MBTL1
SCHEMBL28292577 0.82 CCNC (0.48) MAOBSCN9AL3MBTL1
SCHEMBL28940932 0.81 CNR2 (0.49) MAOBSCN9AMAPTL3MBTL1
SCHEMBL28940985 0.81 SCN9A (0.44) MAOBSCN9A
SCHEMBL28292586 0.81 SCN9A (0.44) MAOBSCN9A
SCHEMBL28284688 0.80 CCNC (0.43) CNR1PDE10AMAPT
SCHEMBL28292579 0.79 CNR2 (0.50) MAOBSCN9ACNR1
SCHEMBL12896110 0.78 KMT2A (0.46) MAOBMMP13CNR1PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN claimed
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed