SCHEMBL28292577

SCHEMBL28292577

CC(C)(O)CNC(=O)c1ccc(OC(N)=O)cn1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCNC P24863 1/20 0.48
CDK8 P49336 1/20 0.48
CDK19 Q9BWU1 1/20 0.48
SCN9A Q15858 4/20 0.47
CNR2 P34972 2/20 0.43
CFTR P13569 1/20 0.42
MAOB P27338 1/20 0.40
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
POLB P06746 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
HPGD P15428 1/20 0.37
CYP2C19 P33261 1/20 0.37
ATM Q13315 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28940932 0.88 CNR2 (0.49) CCNCCDK8CDK19SCN9ACNR2
SCHEMBL28294317 0.87 SCN9A (0.45) CCNCCDK8CDK19SCN9AMAOB
SCHEMBL28940894 0.85 CCNC (0.39) CCNCCDK8CDK19SCN9ACNR2
SCHEMBL28940978 0.83 SCN9A (0.39) CCNCCDK8CDK19SCN9ACNR2
SCHEMBL21379449 0.82 SCN9A (0.44) CCNCCDK8CDK19SCN9ACNR2
SCHEMBL28292566 0.82 MAOB (0.49) SCN9AMAOBL3MBTL1
SCHEMBL28294334 0.80 LOXL2 (0.46) SCN9ACNR2CFTR
SCHEMBL28292586 0.80 SCN9A (0.44) SCN9ACFTRMAOBCYP2C9HPGD
SCHEMBL28940985 0.80 SCN9A (0.44) SCN9ACFTRMAOBCYP2C9HPGD
SCHEMBL28284688 0.80 CCNC (0.43) CCNCCDK8CDK19ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN claimed
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed