SCHEMBL28294317

SCHEMBL28294317

CC(C)(O)CCNC(=O)c1ccc(OC(N)=O)cn1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 3/20 0.45
MAOB P27338 1/20 0.44
CCNC P24863 2/20 0.39
CDK8 P49336 2/20 0.39
CDK19 Q9BWU1 2/20 0.39
HIF1A Q16665 2/20 0.37
CDK9 P50750 1/20 0.37
MAP3K19 Q56UN5 1/20 0.37
HIPK1 Q86Z02 1/20 0.37
HASPIN Q8TF76 1/20 0.37
DYRK1B Q9Y463 1/20 0.37
KMT2A Q03164 1/20 0.37
CYP4F2 P78329 1/20 0.37
CYP4A11 Q02928 1/20 0.37
SCN10A Q9Y5Y9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28292577 0.87 CCNC (0.48) SCN9AMAOBCCNCCDK8CDK19
SCHEMBL28292566 0.85 MAOB (0.49) SCN9AMAOBHIF1A
SCHEMBL28941005 0.84 SCN9A (0.38) SCN9AMAOBCYP4F2CYP4A11
SCHEMBL28292627 0.82 SCN9A (0.41) SCN9AKMT2ACYP4F2CYP4A11
SCHEMBL28940932 0.81 CNR2 (0.49) SCN9AMAOBCCNCCDK8CDK19
SCHEMBL28940894 0.78 CCNC (0.39) SCN9AMAOBCCNCCDK8CDK19
SCHEMBL28940985 0.78 SCN9A (0.44) SCN9AMAOB
SCHEMBL28292586 0.78 SCN9A (0.44) SCN9AMAOB
SCHEMBL28284688 0.78 CCNC (0.43) CCNCCDK8CDK19KMT2A
SCHEMBL22341942 0.74 P4HTM (0.46) MAOBHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN claimed
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed