SCHEMBL28950239

SCHEMBL28950239

FC(F)(F)c1ccc(-c2cnc(Br)nc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 7/20 0.54
TRPV1 Q8NER1 1/20 0.47
CA12 O43570 1/20 0.43
CA9 Q16790 1/20 0.43
SCN2A Q99250 2/20 0.41
MAP4K4 O95819 1/20 0.41
MAOB P27338 2/20 0.40
COMT P21964 1/20 0.40
BACE1 P56817 1/20 0.39
SCN5A Q14524 1/20 0.39
CLK1 P49759 1/20 0.38
KDM1A O60341 1/20 0.38
S1PR1 P21453 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1549633 0.79 KIF11 (0.54) KIF11CA12CA9SCN2A
SCHEMBL11468663 0.79 KIF11 (0.59) KIF11CA12CA9SCN2AMAP4K4
SCHEMBL29818212 0.79 KIF11 (0.59) KIF11MAP4K4MAOBCLK1
SCHEMBL1740256 0.79 KIF11 (0.54) KIF11TRPV1CA12CA9SCN2A
SCHEMBL1549455 0.79 KIF11 (0.48) KIF11TRPV1CA12CA9SCN2A
SCHEMBL11403140 0.77 KMT2A (0.38) KIF11TRPV1MAOB
SCHEMBL197238 0.76 KIF11 (0.78) KIF11MAOB
SCHEMBL29914837 0.76 KIF11 (0.78) KIF11MAOB
SCHEMBL13410633 0.76 KIF11 (0.78) KIF11MAOB
SCHEMBL27642441 0.76 KIF11 (0.46) KIF11TRPV1CA12CA9SCN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115521290-A Preparation of 1, 4-disubstituted indole compound and anti-tumor application thereof 四川大学华西医院 2022-12-27 CN disclosed