SCHEMBL28950487

SCHEMBL28950487

CC(C)(C)OC(=O)CC(O)CCCCCO[Si](c1ccccc1)(c1ccccc1)C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.38
TRPV1 Q8NER1 2/20 0.35
CYP3A4 P08684 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ACACB O00763 1/20 0.33
ACACA Q13085 1/20 0.33
SMYD2 Q9NRG4 2/20 0.33
HDAC4 P56524 2/20 0.33
HDAC1 Q13547 2/20 0.33
ABCB1 P08183 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
AAK1 Q2M2I8 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC10 Q969S8 1/20 0.32
HDAC11 Q96DB2 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28950485 1.00 TRPA1 (0.38) TRPA1TRPV1CYP3A4HTTSMN1; SMN2
SCHEMBL28950526 0.88 GPR84 (0.43) TRPA1TRPV1CYP3A4HTTSMN1; SMN2
SCHEMBL28950527 0.88 GPR84 (0.43) TRPA1TRPV1CYP3A4HTTSMN1; SMN2
SCHEMBL28950596 0.84 CYP3A4 (0.36) CYP3A4HTTSMN1; SMN2SMYD2HDAC4
SCHEMBL17755904 0.84 CYP3A4 (0.35) CYP3A4HTTSMN1; SMN2SMYD2ABCB1
SCHEMBL14254923 0.82 LTB4R (0.37) CYP3A4HTTSMN1; SMN2SMYD2HDAC4
SCHEMBL14315531 0.82 SMYD2 (0.35) CYP3A4HTTSMN1; SMN2SMYD2HDAC1
SCHEMBL14596703 0.81 AAK1 (0.36) CYP3A4HTTSMN1; SMN2SMYD2HDAC4
SCHEMBL29471781 0.81 SMYD2 (0.36) TRPA1CYP3A4HTTSMN1; SMN2ACACB
SCHEMBL29113327 0.81 CSNK1E (0.38) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115551862-A Macrocyclic inhibitors of peptidyl arginine deiminase 吉利德科学公司 2022-12-30 CN disclosed