SCHEMBL28958552

SCHEMBL28958552

CCOC(=O)C1=Nc2ccc(Cl)cc2C1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.48
MAPT P10636 2/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
ALOX15 P16050 7/20 0.43
ALPL P05186 1/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
MAPK10 P53779 1/20 0.41
MAOB P27338 1/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPK1 P28482 1/20 0.40
TRPM8 Q7Z2W7 1/20 0.40
CYP1A2 P05177 1/20 0.40
HPGD P15428 1/20 0.40
XBP1 P17861 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTT P42858 1/20 0.40
TRPV1 Q8NER1 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5639160 0.80 MAPT (0.48) KDM4EMAPTNPC1RAB9AALOX15
SCHEMBL9724293 0.71 GAA (0.43) KDM4EMAPTNPC1RAB9AKMT2A
SCHEMBL29293278 0.70 PDE3B (0.41) KDM4EMAPTKMT2AMEN1ALDH1A1
SCHEMBL7724178 0.69 CA12 (0.48) KDM4EMAPTNPC1RAB9AKMT2A
SCHEMBL549144 0.69 MAPK1 (0.54) KDM4EMAPTALOX15KMT2AMAOB
SCHEMBL7678910 0.69 GAA (0.40) KDM4EMAPTNPC1RAB9AALOX15
SCHEMBL9178589 0.68 MAPT (0.51) KDM4EMAPTNPC1RAB9AKMT2A
SCHEMBL235046 0.67 TSHR (0.60) KDM4EMAPTALOX15KMT2AMAOB
SCHEMBL20774535 0.67 RPS6KA3 (0.48) KDM4EMAPTALOX15ALPLMAOB
SCHEMBL11679386 0.67 MAOB (0.41) KDM4EMAPTNPC1RAB9AALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112920208-B Boric acid-containing indole aryl sulfone derivative and preparation method and application thereof 山东大学 2022-11-08 CN claimed
CN-112920208-B Boric acid-containing indole aryl sulfone derivative and preparation method and application thereof 山东大学 2022-11-08 CN disclosed