SCHEMBL28963147

SCHEMBL28963147

Cc1ccc(-c2nnc(O[C@@H]3CCCN(C(=O)O)C3)c3ccccc23)c(O)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.43
HCRTR2 O43614 2/20 0.43
NLRP3 Q96P20 3/20 0.41
BTK Q06187 1/20 0.39
IL1B P01584 1/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 1/20 0.37
PBRM1 Q86U86 2/20 0.37
MAPT P10636 1/20 0.37
MAPK1 P28482 3/20 0.36
KDM4E B2RXH2 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
RAD52 P43351 1/20 0.35
SMO Q99835 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
USP2 O75604 1/20 0.35
GAA P10253 1/20 0.35
PIK3CD O00329 1/20 0.35
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28963149 1.00 HCRTR1 (0.43) HCRTR1HCRTR2NLRP3BTKIL1B
SCHEMBL28934423 0.88 PIK3CD (0.46) HCRTR1HCRTR2PBRM1PIK3CD
SCHEMBL28934426 0.88 PIK3CD (0.46) HCRTR1HCRTR2PBRM1PIK3CD
SCHEMBL30168040 0.87 NLRP3 (0.52) HCRTR1HCRTR2NLRP3IL1BPBRM1
SCHEMBL30108771 0.87 NLRP3 (0.52) HCRTR1HCRTR2NLRP3IL1BPBRM1
SCHEMBL24840287 0.87 NLRP3 (0.52) HCRTR1HCRTR2NLRP3IL1BPBRM1
SCHEMBL28934400 0.87 NLRP3 (0.52) HCRTR1HCRTR2NLRP3IL1BPBRM1
SCHEMBL29131878 0.86 IL1B (0.42) NLRP3BTKIL1BPBRM1SMO
SCHEMBL29131876 0.86 IL1B (0.42) NLRP3BTKIL1BPBRM1SMO
SCHEMBL28934321 0.80 NLRP3 (0.41) NLRP3BTKIL1BALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115433163-A NLRP3 inflammasome inhibitor and application thereof 药捷安康(南京)科技股份有限公司 2022-12-06 CN disclosed