SCHEMBL29131878

SCHEMBL29131878

O=C(O)N1CCCC(Oc2nnc(-c3ccc(C(F)(F)F)cc3O)c3ccccc23)C1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IL1B P01584 5/20 0.42
NLRP3 Q96P20 5/20 0.41
SMO Q99835 2/20 0.39
LOXL2 Q9Y4K0 3/20 0.38
LOX P28300 1/20 0.38
BTK Q06187 2/20 0.38
KCNH2 Q12809 1/20 0.36
ENPP2 Q13822 3/20 0.36
PBRM1 Q86U86 2/20 0.35
LIPG Q9Y5X9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29131876 1.00 IL1B (0.42) IL1BNLRP3SMOLOXL2LOX
SCHEMBL24925909 0.92 IL1B (0.43) IL1BNLRP3SMOBTKKCNH2
SCHEMBL29131886 0.87 IL1B (0.54) IL1BNLRP3KCNH2
SCHEMBL29275818 0.87 IL1B (0.54) IL1BNLRP3KCNH2
SCHEMBL29131880 0.87 IL1B (0.54) IL1BNLRP3KCNH2
SCHEMBL28963149 0.86 HCRTR1 (0.43) IL1BNLRP3SMOBTKPBRM1
SCHEMBL28963147 0.86 HCRTR1 (0.43) IL1BNLRP3SMOBTKPBRM1
SCHEMBL29131901 0.80 IL1B (0.59) IL1BNLRP3SMOBTKKCNH2
SCHEMBL25403629 0.80 IL1B (0.44) IL1BNLRP3SMOKCNH2LIPG
SCHEMBL29131905 0.80 IL1B (0.59) IL1BNLRP3SMOBTKKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116969920-A Fused pyridazine derivative, preparation method and medical application thereof 上海辉启生物医药科技有限公司 2023-10-31 CN disclosed