SCHEMBL28964918

SCHEMBL28964918

COc1ccc(NS(=O)(=O)c2ccc(Cl)c([N+](=O)[O-])c2)cn1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.67
MEN1 O00255 5/20 0.67
PABPC1 P11940 2/20 0.67
HTT P42858 5/20 0.56
ALDH1A1 P00352 4/20 0.56
LMNA P02545 3/20 0.56
MAPT P10636 2/20 0.56
ALOX15 P16050 2/20 0.56
HPGD P15428 1/20 0.56
MYD88 Q99836 1/20 0.55
VCAM1 P19320 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.53
TSHR P16473 2/20 0.53
USP2 O75604 1/20 0.53
TP53 P04637 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
POLB P06746 2/20 0.53
HSPD1 P10809 2/20 0.49
PTPN2 P17706 2/20 0.49
PTPN1 P18031 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30205653 1.00 KMT2A (0.67) KMT2AMEN1PABPC1HTTALDH1A1
SCHEMBL6677229 0.82 VCAM1 (0.60) KMT2AMEN1ALDH1A1LMNAMAPT
SCHEMBL6678848 0.80 LMNA (0.67) KMT2AMEN1HTTALDH1A1LMNA
SCHEMBL28746841 0.79 ALDH1A1 (0.60) ALDH1A1LMNAHPGDVCAM1SMN1; SMN2
SCHEMBL15544374 0.78 MEN1 (0.62) KMT2AMEN1PABPC1HTTALDH1A1
SCHEMBL5225915 0.78 VCAM1 (0.64) HTTALDH1A1LMNAMAPTVCAM1
SCHEMBL5228187 0.78 VCAM1 (0.64) KMT2AMEN1HTTLMNAMAPT
SCHEMBL6675755 0.77 ALDH1A1 (0.64) KMT2AMEN1HTTALDH1A1LMNA
SCHEMBL6681330 0.77 ALDH1A1 (0.59) KMT2AMEN1HTTALDH1A1LMNA
SCHEMBL27793353 0.77 VCAM1 (0.54) HTTALDH1A1LMNAVCAM1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115710251-B Medullary differentiation factor 88 inhibitor and preparation method and application thereof 杭州医学院 2024-05-28 CN disclosed
CN-115710251-A Myeloid differentiation factor 88 inhibitor and preparation method and application thereof 杭州医学院 2023-02-24 CN disclosed