SCHEMBL28970511

SCHEMBL28970511

NN1C=Cc2ccccc2C1Br

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.44
BRD4 O60885 1/20 0.40
CCL2 P13500 1/20 0.40
HTR6 P50406 1/20 0.35
ATM Q13315 1/20 0.34
KDM4E B2RXH2 2/20 0.33
CYP2D6 P10635 2/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
CHRM2 P08172 1/20 0.33
CYP3A4 P08684 1/20 0.33
CHRM1 P11229 1/20 0.33
DRD2 P14416 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
NFKB1 P19838 1/20 0.33
CHRM3 P20309 1/20 0.33
SLC6A2 P23975 1/20 0.33
HTR2C P28335 1/20 0.33
ADRA1A P35348 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24061842 0.78 BRD4 (0.49) HTR2ABRD4CCL2ATMKDM4E
SCHEMBL28310354 0.69 ALDH1A1 (0.39) HTR2ABRD4CCL2ATMLMNA
SCHEMBL28374476 0.69 BRD4 (0.41) HTR2ABRD4CCL2ATMKDM4E
SCHEMBL28323510 0.68 PRCP (0.35) HTR2ABRD4CCL2ATMDRD2
SCHEMBL7551620 0.65 BRD4 (0.49) HTR2ABRD4CCL2HTR6ATM
SCHEMBL16872444 0.65 CNR2 (0.41) HTR2ABRD4CCL2CYP2D6KCNH2
SCHEMBL31046607 0.64 HTR2A (0.43) HTR2ABRD4CCL2HTR6KDM4E
SCHEMBL6233907 0.64 HTR2A (0.43) HTR2ABRD4CCL2HTR6KDM4E
SCHEMBL10694747 0.63 BRD4 (0.55) HTR2ABRD4CCL2ATMKDM4E
SCHEMBL8256345 0.63 HTR2A (0.69) HTR2ABRD4CCL2HTR6KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114685532-A Macrocyclic compound and medical application thereof 正大天晴药业集团股份有限公司 2022-07-01 CN disclosed