SCHEMBL6233907

SCHEMBL6233907

BrC1C=Cc2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.43
HTR6 P50406 1/20 0.41
KDM4E B2RXH2 3/20 0.34
CYP2D6 P10635 3/20 0.34
TP53 P04637 2/20 0.34
CYP3A4 P08684 2/20 0.34
HSD17B10 Q99714 2/20 0.34
BRD4 O60885 1/20 0.34
CCL2 P13500 1/20 0.34
LMNA P02545 1/20 0.34
CHRM2 P08172 1/20 0.34
CHRM1 P11229 1/20 0.34
DRD2 P14416 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
NFKB1 P19838 1/20 0.34
CHRM3 P20309 1/20 0.34
SLC6A2 P23975 1/20 0.34
HTR2C P28335 1/20 0.34
ADRA1A P35348 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31046607 1.00 HTR2A (0.43) HTR2AHTR6KDM4ECYP2D6TP53
SCHEMBL23100802 0.80 HTR2A (0.36) HTR2AHTR6KDM4ECYP2D6TP53
SCHEMBL25218430 0.78 HTR2A (0.39) HTR2AHTR6KDM4ECYP2D6TP53
SCHEMBL3246033 0.78 HTR2A (0.35) HTR2AHTR6KDM4ECYP2D6BRD4
SCHEMBL8732534 0.77 HTR2A (0.38) HTR2AHTR6KDM4ECYP2D6TP53
SCHEMBL9309445 0.77 HTR2A (0.38) HTR2AHTR6KDM4ECYP2D6TP53
SCHEMBL31068436 0.77 HTR6 (0.41) HTR2AHTR6KDM4ECYP2D6TP53
SCHEMBL8380997 0.77 HTR2A (0.38) HTR2AHTR6KDM4ECYP2D6TP53
SCHEMBL8380915 0.77 HTR2A (0.38) HTR2AHTR6KDM4ECYP2D6TP53
SCHEMBL8383845 0.77 HTR2A (0.38) HTR2AHTR6KDM4ECYP2D6TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 36 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115057831-B Thiadiazole compound and application thereof in preparation of KKBC 1 protein inhibitor 中国医科大学附属盛京医院 2023-08-04 CN claimed
CN-115057831-A Thiadiazole compound and application thereof in preparation of KKLC1 protein inhibitor 中国医科大学附属盛京医院 2022-09-16 CN claimed
CN-1307064-A Monocyclopentadienes catalyst for polymerization of olefin and preparaing method thereof CHINESE ACAD INST CHEMISTRY (CN) 2001-08-08 CN claimed
CN-115362151-B Arylpiperidines as monoacylglycerol lipase modulators 詹森药业有限公司 2025-02-11 CN disclosed
US-20240092781-A1 ARYL PIPERIDINES AS MONOACYLGLYCEROL LIPASE MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2024-03-21 US disclosed
US-11787798-B2 Aryl piperidines as monoacylglycerol lipase modulators JANSSEN PHARMACEUTICA NV (BE) 2023-10-17 US disclosed
CN-111630083-B Polyamide composition comprising specific copolyamide containing caprolactam monomer, semi-crystalline polyamide and reinforcing filler 巴斯夫欧洲公司 2023-09-01 CN disclosed
CN-115612271-B Heat-resistant flame-retardant PC (polycarbonate) reinforced material and production method thereof 江苏松上科技有限公司 2023-08-08 CN disclosed
CN-115057831-B Thiadiazole compound and application thereof in preparation of KKBC 1 protein inhibitor 中国医科大学附属盛京医院 2023-08-04 CN disclosed
CN-114262492-B Heat-resistant flame-retardant ABS material and production method thereof 江苏松上科技有限公司 2023-04-11 CN disclosed
CN-115612271-A Heat-resistant flame-retardant PC (polycarbonate) reinforced material and production method thereof 江苏松上科技有限公司 2023-01-17 CN disclosed
CN-103022376-A Organic light-emitting diode (OLED) device KUNSHAN VISIONOX DISPLAY TECH 2013-04-03 CN disclosed
CN-102010353-A New method for preparing rasagiline mesylate WINCHEM SCIENCE AND TECHNOLOGY CO LTD 2011-04-13 CN disclosed
CN-101381314-A Preparation method of (R)-(+)-N-propargyl-1-indan amines CHENGDU HEALTHCARE PHARMACEUTI (CN) 2009-03-11 CN disclosed
US-6936636-B2 5-[phenyl-tetrahydronaphthalene-2-yl dihydronaphthalen-2-yl and heteroaryl-cyclopropyl]-pentadienoic acid derivatives having serum glucose reducing activity ALLERGAN, INC. (US) 2005-08-30 US disclosed
CN-1653021-A Preparation of substituted indenes BASELL POLYOLEFINE GMBH (DE) 2005-08-10 CN disclosed
WO-2005000784-A2 5-[PHENYL, TETRAHYDRONAPHTHALENE-2-YL DIHYDRONAPHTHALEN-2-YL AND HETEROARYL- CYCLOPROPYL]-PENTADIENOIC ACID DERIVATIVES HAVING SERUM GLUCOSE REDUCING ACTIVITY ALLERGAN, INC. (US) 2005-01-06 WO disclosed
US-20050004213-A1 5-[phenyl-tetrahydronaphthalene-2-yl dihydronaphthalen-2-yl and heteroaryl-cyclopropyl]-pentadienoic acid derivatives having serum glucose reducing activity ALLERGAN, INC. 2005-01-06 US disclosed
CN-1307064-A Monocyclopentadienes catalyst for polymerization of olefin and preparaing method thereof CHINESE ACAD INST CHEMISTRY (CN) 2001-08-08 CN disclosed
EP-0258096-A2 Indane derivatives, process for their preparation, their use as medicines, pharmaceutical compositions containing them and the intermediates obtained ROUSSEL-UCLAF (FR) 1988-03-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240092781-A1 ARYL PIPERIDINES AS MONOACYLGLYCEROL LIPASE MODULATORS MGLL, LPL, PNLIP HTR2A 26/4885HTR6 281/4885KDM4E 1995/4885
US-11787798-B2 Aryl piperidines as monoacylglycerol lipase modulators MGLL, LPL, PNLIP HTR2A 26/4885HTR6 281/4885KDM4E 1995/4885
US-20050004213-A1 5-[phenyl-tetrahydronaphthalene-2-yl dihydronaphthalen-2-yl and heteroaryl-cyclopropyl]-pentadienoic acid derivatives having serum glucose reducing activity PNLIP, TPO, MTTP HTR2A 1227/4885HTR6 1480/4885KDM4E 3712/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.