SCHEMBL28972777

SCHEMBL28972777

COc1ccccc1N1CCN(CCCc2ccccc2C(N)=O)CC1

nearest known ligand 0.67

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.67
HTR7 P34969 4/20 0.67
KDM4E B2RXH2 1/20 0.61
ALDH1A1 P00352 1/20 0.61
TDP1 Q9NUW8 1/20 0.61
DRD2 P14416 4/20 0.59
DRD3 P35462 1/20 0.59
HTR2A P28223 1/20 0.58
DRD4 P21917 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8980582 0.92 HTR1A (0.62) HTR1AHTR7KDM4EALDH1A1TDP1
SCHEMBL27454683 0.90 KDM4E (0.65) HTR1AHTR7KDM4EALDH1A1TDP1
Hydrochloric Acid SCHEMBL27508537 0.89 KDM4E (0.64) HTR1AHTR7KDM4EALDH1A1TDP1
SCHEMBL27455347 0.85 MEN1 (0.60) HTR1AHTR7KDM4EALDH1A1TDP1
SCHEMBL3188003 0.82 ALDH1A1 (0.71) HTR1AHTR7KDM4EALDH1A1TDP1
SCHEMBL11446717 0.82 HTR1A (0.75) HTR1AHTR7DRD2DRD3DRD4
Hydrochloric Acid SCHEMBL3196115 0.81 HTR1A (0.71) HTR1AHTR7KDM4EALDH1A1TDP1
SCHEMBL6956822 0.81 KDM4E (0.72) HTR1AHTR7KDM4EALDH1A1TDP1
SCHEMBL28972654 0.80 DRD2 (0.58) HTR1AHTR7DRD2DRD3HTR2A
SCHEMBL27470893 0.80 DRD2 (0.59) HTR1AHTR7KDM4EALDH1A1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110511215-B Aryl piperazine/piperidine compound and application thereof 复旦大学 2023-03-28 CN disclosed