SCHEMBL28973006

SCHEMBL28973006

COc1nc(N2CCOCC2)c([N+](=O)[O-])cc1NC(C)=O

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.45
MAPT P10636 7/20 0.43
HTT P42858 1/20 0.42
MAPK1 P28482 2/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
RAB9A P51151 1/20 0.41
POLB P06746 1/20 0.40
PKM P14618 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24251673 0.90 ALDH1A1 (0.44) ALDH1A1MAPTHTTMAPK1KMT2A
SCHEMBL28973016 0.86 MAPT (0.39) ALDH1A1MAPTMAPK1KMT2ASMN1; SMN2
SCHEMBL28510516 0.85 ALDH1A1 (0.44) ALDH1A1MAPTMAPK1SMN1; SMN2LMNA
SCHEMBL29133298 0.80 WDR5 (0.43) ALDH1A1MAPTMAPK1SMN1; SMN2LMNA
SCHEMBL27238331 0.80 WDR5 (0.43) ALDH1A1MAPTMAPK1SMN1; SMN2LMNA
SCHEMBL10745494 0.78 POLB (0.49) ALDH1A1MAPTHTTKMT2ASMN1; SMN2
SCHEMBL28973031 0.78 MAPT (0.35) ALDH1A1MAPTHTTMAPK1KMT2A
SCHEMBL17490464 0.78 NPSR1 (0.46) ALDH1A1MAPTHTTKMT2ASMN1; SMN2
SCHEMBL28973029 0.77 MCHR1 (0.38) ALDH1A1MAPTMAPK1SMN1; SMN2LMNA
SCHEMBL28359061 0.76 WDR5 (0.40) ALDH1A1MAPTMAPK1SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115701429-B 4- (1H-indol-1-yl) pyrimidine-2-amino derivative, and preparation method and application thereof 上海和誉生物医药科技有限公司 2024-03-12 CN disclosed
CN-115701429-A 4- (1H-indole-1-yl) pyrimidine-2-amino derivative and preparation method and application thereof 上海和誉生物医药科技有限公司 2023-02-10 CN disclosed