SCHEMBL24251673

SCHEMBL24251673

COc1nc(N2CCCC2)c([N+](=O)[O-])cc1NC(C)=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.44
MAPK1 P28482 3/20 0.44
HTT P42858 1/20 0.44
MAPT P10636 10/20 0.43
POLB P06746 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
NPSR1 Q6W5P4 3/20 0.41
LMNA P02545 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
GALR2 O43603 1/20 0.41
MITF O75030 1/20 0.41
HSP90AA1 P07900 1/20 0.41
HPGD P15428 1/20 0.41
XBP1 P17861 1/20 0.41
CCR6 P51684 1/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
OPRK1 P41145 1/20 0.40
ALOX12 P18054 1/20 0.38
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28973006 0.90 ALDH1A1 (0.45) ALDH1A1MAPK1HTTMAPTPOLB
SCHEMBL24251711 0.84 ALDH1A1 (0.41) ALDH1A1MAPK1HTTMAPTPOLB
SCHEMBL27238331 0.82 WDR5 (0.43) ALDH1A1MAPK1MAPTPOLBTDP1
SCHEMBL29133298 0.82 WDR5 (0.43) ALDH1A1MAPK1MAPTPOLBTDP1
SCHEMBL10745494 0.81 POLB (0.49) ALDH1A1HTTMAPTPOLBNPSR1
SCHEMBL17490464 0.80 NPSR1 (0.46) ALDH1A1HTTMAPTPOLBNPSR1
SCHEMBL27238138 0.79 MAPT (0.36) ALDH1A1MAPTPOLBNPSR1LMNA
SCHEMBL27238175 0.79 MAPT (0.36) ALDH1A1MAPTPOLBNPSR1LMNA
SCHEMBL28359061 0.78 WDR5 (0.40) ALDH1A1MAPK1MAPTPOLBNPSR1
SCHEMBL24251657 0.78 ALDH1A1 (0.49) ALDH1A1MAPK1HTTMAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022033455-A1 TRIAZINE DERIVATIVE HAVING EGFR INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 上海和誉生物医药科技有限公司 2022-02-17 WO disclosed