SCHEMBL28974587

SCHEMBL28974587

CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)Nc1ccc2[nH]c(C(=O)O)cc2c1

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.54
F11 P03951 9/20 0.53
CTSS P25774 4/20 0.53
CTSK P43235 3/20 0.53
CTSB P07858 2/20 0.53
CTSL P07711 1/20 0.53
PYGL P06737 3/20 0.52
ACE P12821 1/20 0.48
AKT1 P31749 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28974589 1.00 HDAC8 (0.54) HDAC8F11CTSSCTSKCTSB
SCHEMBL28602428 0.92 F11 (0.55) HDAC8F11CTSSCTSK
SCHEMBL28919287 0.92 F11 (0.55) HDAC8F11CTSSCTSK
SCHEMBL23466599 0.90 MMP13 (0.55) HDAC8F11CTSSCTSKCTSB
SCHEMBL23466603 0.90 MMP13 (0.55) HDAC8F11CTSSCTSKCTSB
SCHEMBL29758100 0.90 MMP13 (0.55) HDAC8F11CTSSCTSKCTSB
SCHEMBL28673878 0.88 KLK7 (0.46) HDAC8F11CTSS
SCHEMBL28673880 0.88 KLK7 (0.46) HDAC8F11CTSS
SCHEMBL28692985 0.88 F11 (0.45) HDAC8F11CTSSCTSKCTSB
SCHEMBL28692986 0.88 F11 (0.45) HDAC8F11CTSSCTSKCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114728917-A Oxamide derivative, preparation method and medical application thereof 深圳信立泰药业股份有限公司 2022-07-08 CN disclosed