SCHEMBL28975596

SCHEMBL28975596

CC(C)(C)OC(=O)NCc1nnc(-c2ccc(CC(=O)O)cc2)nn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.46
EPHX2 P34913 1/20 0.42
NR1H4 Q96RI1 1/20 0.42
NAMPT P43490 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
RXRA P19793 2/20 0.40
RXRB P28702 2/20 0.40
RXRG P48443 2/20 0.40
GLS O94925 3/20 0.40
SDCBP O00560 1/20 0.39
SDC2 P34741 1/20 0.39
CYP17A1 P05093 1/20 0.39
GRM2 Q14416 1/20 0.39
HDAC6 Q9UBN7 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
ATR Q13535 1/20 0.38
ABCC4 O15439 1/20 0.38
LMNA P02545 1/20 0.38
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25497278 0.86 HDAC1 (0.47) HDAC1NAMPTGLSCTSSCTSK
SCHEMBL26328902 0.85 MAPT (0.42) HDAC1NAMPTL3MBTL1LMNAAKT1
SCHEMBL26328906 0.84 NAMPT (0.41) HDAC1EPHX2NR1H4NAMPTL3MBTL1
SCHEMBL30736827 0.83 HDAC1 (0.58) HDAC1EPHX2NR1H4NAMPTL3MBTL1
SCHEMBL25439945 0.82 NAMPT (0.41) HDAC1NAMPTL3MBTL1HDAC6ATR
SCHEMBL26329031 0.82 DYRK1A (0.44) EPHX2NR1H4L3MBTL1LMNATSHR
SCHEMBL1244728 0.81 EPHX2 (0.56) HDAC1EPHX2NR1H4NAMPTL3MBTL1
SCHEMBL25367309 0.81 NAMPT (0.47) HDAC1NAMPTL3MBTL1GLSSDCBP
SCHEMBL15322811 0.80 NAMPT (0.50) HDAC1NAMPTL3MBTL1SDCBPSDC2
SCHEMBL13977598 0.78 KDM4E (0.49) NAMPTL3MBTL1LMNAGAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115873014-B Controllable proteolytic targeted chimera and application thereof 中国药科大学 2024-08-20 CN disclosed
CN-115991880-B Dendrimer PAMAM-G5-TCO and preparation method and application thereof 中国药科大学 2024-03-19 CN disclosed
CN-115991880-A Dendrimer PAMAM-G5-TCO and preparation method and application thereof 中国药科大学 2023-04-21 CN disclosed
CN-115873014-A Controllable proteolysis targeting chimera and application thereof 中国药科大学 2023-03-31 CN disclosed