SCHEMBL2898301

SCHEMBL2898301

COc1cccc2c1C(Nc1ccc3c(NS(=O)(=O)C4=CC=CC(F)(F)C4)cccc3n1)CC2

nearest known ligand 0.31

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.31
HTR1A P08908 1/20 0.31
MCHR1 Q99705 1/20 0.30
PFKFB3 Q16875 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1616695 0.82 ALDH1A1 (0.42) KDM4E
SCHEMBL1616597 0.81 MAP2K4 (0.38) KDM4EPFKFB3
SCHEMBL1615349 0.80 MAP2K4 (0.38) KDM4EPFKFB3
SCHEMBL2243192 0.80 ACHE (0.42) KDM4EHTR1AMCHR1PFKFB3
SCHEMBL1615734 0.77 PFKFB3 (0.39) KDM4EPFKFB3
SCHEMBL1615961 0.76 KDM4E (0.34) KDM4EMCHR1
SCHEMBL2905912 0.73 MCHR1 (0.39) HTR1AMCHR1PFKFB3
SCHEMBL1615706 0.72 METAP2 (0.38) KDM4E
SCHEMBL2243251 0.71 MEN1 (0.41)
SCHEMBL1615576 0.70 CA1 (0.38) KDM4EPFKFB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099763-B1 2-AMINOQUINOLINES AS 5-HT(5A) RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-08-11 EP claimed