SCHEMBL28985187

SCHEMBL28985187

COc1ccnc(C(C)C=Cc2ccccc2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.44
CYP1A1 P04798 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP1B1 Q16678 2/20 0.42
CCR1 P32246 1/20 0.41
CCR5 P51681 1/20 0.41
CCR8 P51685 1/20 0.41
CYP3A4 P08684 2/20 0.41
MAPT P10636 2/20 0.41
KDM4E B2RXH2 2/20 0.41
HPGD P15428 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MEN1 O00255 1/20 0.41
USP2 O75604 1/20 0.41
ALDH1A1 P00352 1/20 0.41
TP53 P04637 1/20 0.41
KMT2A Q03164 1/20 0.41
TRPV1 Q8NER1 1/20 0.41
HSD17B10 Q99714 1/20 0.41
NFE2L2 Q16236 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28985184 1.00 TRPA1 (0.44) TRPA1CYP1A1CYP1A2CYP1B1CCR1
SCHEMBL28985179 0.84 LCK (0.49) CYP1A1CYP1A2CYP3A4KDM4ESMN1; SMN2
SCHEMBL28985175 0.84 LCK (0.49) CYP1A1CYP1A2CYP3A4KDM4ESMN1; SMN2
SCHEMBL28985162 0.81 GRM4 (0.41) CCR1CCR5CCR8KDM4EHPGD
SCHEMBL28985163 0.81 GRM4 (0.41) CCR1CCR5CCR8KDM4EHPGD
SCHEMBL28985307 0.77 RELA (0.44) CYP1B1MAPTKDM4ESMN1; SMN2MEN1
SCHEMBL28985306 0.77 SLC6A2 (0.44) CYP1A2CYP3A4MAPTKDM4EMEN1
SCHEMBL28985305 0.77 SLC6A2 (0.44) CYP1A2CYP3A4MAPTKDM4EMEN1
SCHEMBL29000588 0.74 TRPA1 (0.55) TRPA1CYP1A1CYP1A2CYP1B1CCR1
SCHEMBL5664369 0.73 NOS3 (0.55) CCR1CCR5CCR8NOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115974927-A Diamine-derived phosphine chiral phosphine oxide ligand-promoted nickel-catalyzed asymmetric alkylation of pyridine C2-H bond 南开大学 2023-04-18 CN disclosed