SCHEMBL28985437

SCHEMBL28985437

O=C(O)N1CCC=C(c2ccncc2)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MYC P01106 2/20 0.39
ALDH1A1 P00352 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
GRM5 P41594 1/20 0.36
NAMPT P43490 1/20 0.34
PDE10A Q9Y233 2/20 0.34
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 2/20 0.33
CYP2C9 P11712 1/20 0.33
ROCK2 O75116 1/20 0.33
ROCK1 Q13464 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA7 P36544 1/20 0.33
CHRNA4 P43681 1/20 0.33
FNTA P49354 1/20 0.33
FNTB P49356 1/20 0.33
NAPRT Q6XQN6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15140927 0.85 ALDH1A1 (0.42) MYCALDH1A1SMN1; SMN2KMT2AMEN1
SCHEMBL29640885 0.82 MYC (0.43) MYCALDH1A1KMT2AHSD17B10MEN1
SCHEMBL28985440 0.82 MKNK1 (0.42) MYCALDH1A1CYP2C9
SCHEMBL28369802 0.81 MYC (0.34) MYCCHRNB2CHRNA4
SCHEMBL31450581 0.81 LSS (0.46) MYCALDH1A1SMN1; SMN2NAMPTCHRNB2
SCHEMBL28539765 0.80 MEN1 (0.41) MYCNAMPTKMT2ACYP2C9MEN1
SCHEMBL22441484 0.79 GRM1 (0.48) GRM5NAMPTPDE10A
SCHEMBL21193344 0.77 HCAR2 (0.35) MYC
SCHEMBL1856104 0.75 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2NAMPTKMT2AKDM4E
SCHEMBL25243642 0.75 CHRNB2 (0.62) MYCALDH1A1PDE10AKMT2AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116390917-A MRGX2 antagonists 葛兰素史密斯克莱知识产权发展有限公司 2023-07-04 CN disclosed
CN-110818683-B 2-pyridine substituted urea structure small molecule compound and synthesis and application thereof 中国科学院上海药物研究所 2023-04-14 CN disclosed