SCHEMBL2898934

SCHEMBL2898934

O=C(/C=C/c1ccc(F)c(Cl)c1)N1CCC(=O)N(CCCCN2CCCC(CO)C2)CC1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PYGL P06737 2/20 0.43
CCR2 P41597 4/20 0.42
GPR183 P32249 3/20 0.41
ITGB2 P05107 2/20 0.39
ICAM1 P05362 2/20 0.39
ITGAL P20701 2/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2896881 0.93 CCR2 (0.47) PYGLCCR2GPR183
SCHEMBL2902759 0.92 PYGL (0.42) PYGLCCR2GPR183ITGB2ICAM1
SCHEMBL2899943 0.91 CCR2 (0.47) PYGLCCR2GPR183
SCHEMBL2905026 0.90 PYGL (0.44) PYGLCCR2GPR183ITGB2ICAM1
SCHEMBL2922190 0.90 CCR2 (0.50) PYGLCCR2GPR183MEN1KMT2A
SCHEMBL2922192 0.90 CCR2 (0.50) PYGLCCR2GPR183MEN1KMT2A
SCHEMBL2904266 0.89 PYGL (0.42) PYGLCCR2GPR183ITGB2ICAM1
SCHEMBL2904263 0.89 PYGL (0.42) PYGLCCR2GPR183ITGB2ICAM1
SCHEMBL2904260 0.89 PYGL (0.42) PYGLCCR2GPR183ITGB2ICAM1
SCHEMBL2899254 0.89 CCR2 (0.50) PYGLCCR2GPR183MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010506-B1 DIAZEPAN DERIVATIVES MODULATORS OF CHEMOKINE RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-04 EP disclosed