SCHEMBL2904263

SCHEMBL2904263

O=C(C=Cc1ccc(F)c(Cl)c1)N1CCC(=O)N(CCCN2CCCC(O)C2)CC1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PYGL P06737 2/20 0.42
GPR183 P32249 4/20 0.42
CCR2 P41597 3/20 0.41
ITGB2 P05107 2/20 0.40
ICAM1 P05362 2/20 0.40
ITGAL P20701 2/20 0.40
CYP2C19 P33261 2/20 0.39
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP2D6 P10635 1/20 0.38
ATM Q13315 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2904266 1.00 PYGL (0.42) PYGLGPR183CCR2ITGB2ICAM1
SCHEMBL2904260 1.00 PYGL (0.42) PYGLGPR183CCR2ITGB2ICAM1
SCHEMBL2905026 0.98 PYGL (0.44) PYGLGPR183CCR2ITGB2ICAM1
SCHEMBL2904597 0.93 CCR2 (0.44) PYGLGPR183CCR2ITGB2ICAM1
SCHEMBL2902431 0.93 GPR183 (0.48) PYGLGPR183CCR2
SCHEMBL2902199 0.93 GPR183 (0.48) PYGLGPR183CCR2
SCHEMBL2902196 0.93 GPR183 (0.48) PYGLGPR183CCR2
SCHEMBL2902434 0.93 GPR183 (0.48) PYGLGPR183CCR2
SCHEMBL2902201 0.93 GPR183 (0.48) PYGLGPR183CCR2
SCHEMBL4243628 0.93 GPR183 (0.48) PYGLGPR183CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010506-B1 DIAZEPAN DERIVATIVES MODULATORS OF CHEMOKINE RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-04 EP disclosed