SCHEMBL28989529

SCHEMBL28989529

O=C(O)c1cc(B(O)O)ccc1Br

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.41
CA1 P00915 3/20 0.41
CA2 P00918 3/20 0.41
TSHR P16473 2/20 0.41
LCK P06239 1/20 0.40
FYN P06241 1/20 0.40
CA12 O43570 1/20 0.39
CA3 P07451 1/20 0.39
CA4 P22748 1/20 0.39
CA6 P23280 1/20 0.39
CA5A P35218 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA13 Q8N1Q1 1/20 0.39
CA14 Q9ULX7 1/20 0.39
CA5B Q9Y2D0 1/20 0.39
AKR1C4 P17516 2/20 0.38
AKR1C3 P42330 2/20 0.38
AKR1C2 P52895 2/20 0.38
AKR1C1 Q04828 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30807652 0.81 ALDH1A1 (0.44) HSD17B10CA1CA2TSHRCA12
SCHEMBL918043 0.81 ALDH1A1 (0.44) HSD17B10CA1CA2TSHRCA12
SCHEMBL18593627 0.78 TTBK1 (0.40) HSD17B10CA1CA2TSHRCA12
SCHEMBL733036 0.76 KDM4E (0.44) CA1CA2AKR1C2AKR1C1KDM4E
SCHEMBL18241272 0.76 CA2 (0.41) HSD17B10CA2TSHRKDM4E
SCHEMBL787718 0.76 ALDH1A1 (0.59) TSHRKDM4ESMN1; SMN2TTRCTDSP1
SCHEMBL29825352 0.76 KDM4E (0.44) CA1CA2AKR1C2AKR1C1KDM4E
SCHEMBL29954641 0.76 ALDH1A1 (0.59) TSHRKDM4ESMN1; SMN2TTRCTDSP1
SCHEMBL1163265 0.76 KDM4E (0.50) HSD17B10CA1CA2LCKFYN
SCHEMBL29955154 0.76 KDM4E (0.50) HSD17B10CA1CA2LCKFYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115996932-A New macrocyclic LRRK2 kinase inhibitors 法国施维雅药厂 2023-04-21 CN disclosed