SCHEMBL28989690

SCHEMBL28989690

CC(C)(C)OC(=O)NC(Cc1ccc(Br)s1)C(N)=O

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSS P25774 11/20 0.44
CTSK P43235 10/20 0.44
REN P00797 3/20 0.44
AAK1 Q2M2I8 2/20 0.41
CTSB P07858 2/20 0.40
CTSL P07711 2/20 0.40
ACE P12821 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
SCN9A Q15858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16065010 1.00 CTSS (0.44) CTSSCTSKRENAAK1CTSB
SCHEMBL539422 0.89 ACE (0.50) CTSSCTSKCTSBCTSLACE
SCHEMBL3376657 0.89 ACE (0.50) CTSSCTSKCTSBCTSLACE
SCHEMBL4245453 0.88 KLK5 (0.46) CTSSCTSKAAK1CTSBCTSL
SCHEMBL539352 0.88 KLK5 (0.46) CTSSCTSKAAK1CTSBCTSL
SCHEMBL539351 0.88 KLK5 (0.46) CTSSCTSKAAK1CTSBCTSL
SCHEMBL24981557 0.79 CTSS (0.46) CTSSCTSKCTSBCTSL
SCHEMBL28989397 0.79 CTSS (0.46) CTSSCTSKCTSBCTSL
SCHEMBL9109956 0.79 CTSK (0.68) CTSSCTSKRENCTSBCTSL
SCHEMBL9109963 0.79 CTSK (0.68) CTSSCTSKRENCTSBCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115996923-A Nitrile derivative as dipeptidyl peptidase 1 inhibitor and application thereof 四川海思科制药有限公司 2023-04-21 CN disclosed