SCHEMBL2899052

SCHEMBL2899052

Cc1cc(Cl)cc(C(=O)NC2CSC2)c1C(N)=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.40
RAB9A P51151 6/20 0.40
POLB P06746 2/20 0.39
TAS1R3 Q7RTX0 2/20 0.38
TAS1R1 Q7RTX1 2/20 0.38
TAS1R2 Q8TE23 2/20 0.38
HPGD P15428 2/20 0.36
ALDH1A1 P00352 2/20 0.36
CHEK1 O14757 1/20 0.35
P2RX7 Q99572 1/20 0.35
KDM4E B2RXH2 1/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
NFKB1 P19838 1/20 0.34
MAPK1 P28482 1/20 0.34
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2899055 0.85 NPC1 (0.41) NPC1RAB9APOLBTAS1R3TAS1R1
SCHEMBL2901313 0.83 POLB (0.37) NPC1RAB9APOLBTAS1R3TAS1R1
SCHEMBL4666210 0.78 POLB (0.45) NPC1RAB9APOLBHPGDALDH1A1
SCHEMBL2900855 0.76 POLB (0.36) NPC1RAB9APOLBHPGDALDH1A1
SCHEMBL14697697 0.76 POLB (0.42) NPC1RAB9APOLBHPGDALDH1A1
SCHEMBL2783255 0.75 CHRM1 (0.43) POLB
SCHEMBL2786923 0.74 POLB (0.41) NPC1RAB9APOLBHPGDALDH1A1
SCHEMBL2695475 0.74 NPC1 (0.48) NPC1RAB9APOLBP2RX7
SCHEMBL4639194 0.72 POLB (0.59) RAB9APOLBHPGDALDH1A1KDM4E
SCHEMBL27779125 0.71 ALDH1A1 (0.48) NPC1RAB9APOLBTAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2213167-B1 Anthranilamide derivatives and their use for the control of insects and acari SYNGENTA PARTICIPATIONS AG (CH) 2013-07-31 EP disclosed
US-8278464-B2 Insecticides SYNGENTA CROP PROTECTION LLC (US) 2012-10-02 US disclosed
US-8084474-B2 Insecticides SYNGENTA CROP PROTECTION, INC. (US) 2011-12-27 US disclosed
EP-2213167-A1 Anthranilamide derivatives and their use for the control of insects and acari Syngenta Participations AG (CH) 2010-08-04 EP disclosed
US-20100168066-A1 NOVEL INSECTICIDES SYNGENTA CROP PROTECTION, INC. (US) 2010-07-01 US disclosed
EP-1976385-A2 ANTHRANILAMIDE DERIVATIVES AND THEIR USE FOR THE CONTROL OF INSECTS AND ACARI Syngeta Participations AG (CH) 2008-10-08 EP disclosed
WO-2007080131-A2 ANTHRANILAMIDE DERIVATIVES AND THEIR USE FOR THE CONTROL OF INSECTS AND ACARI SYNGENTA PARTICIPATIONS AG (CH) 2007-07-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100168066-A1 NOVEL INSECTICIDES DDT, ACHE, CYP4F11 NPC1 1329/4885RAB9A 738/4885POLB 4402/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.