SCHEMBL28990876

SCHEMBL28990876

c1coc(-n2ccc(N3CCNCC3)n2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLD1 Q13393 1/20 0.41
HTR3E A5X5Y0 3/20 0.39
HTR3B O95264 3/20 0.39
HTR3A P46098 3/20 0.39
HTR3D Q70Z44 3/20 0.39
HTR3C Q8WXA8 3/20 0.39
ALDH1A1 P00352 2/20 0.39
ADRB1 P08588 4/20 0.38
HTR2C P28335 2/20 0.38
HRH3 Q9Y5N1 2/20 0.38
KDM4E B2RXH2 1/20 0.38
USP2 O75604 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
HTR1A P08908 1/20 0.38
MAPK1 P28482 1/20 0.38
SLC6A4 P31645 1/20 0.38
HTR7 P34969 1/20 0.38
HTT P42858 1/20 0.38
HTR6 P50406 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5029237 0.77 ADRB1 (0.47) PLD1HTR3EHTR3BHTR3AHTR3D
SCHEMBL3629025 0.75 ADRB1 (0.56) PLD1HTR3EHTR3BHTR3AHTR3D
SCHEMBL20458913 0.71 CHRNB2 (0.45) HTR3EHTR3BHTR3AHTR3DHTR3C
Pyridine SCHEMBL27687558 0.71 PLD1 (0.47) PLD1HTR3EHTR3BHTR3AHTR3D
SCHEMBL27538736 0.71 ADRB1 (0.39) PLD1HTR3EHTR3BHTR3AHTR3D
SCHEMBL30411053 0.69 HRH3 (0.73) PLD1ADRB1HRH3CYP1A2HSD17B10
SCHEMBL29691124 0.68 HTR2C (0.47) PLD1ADRB1HTR2CKDM4ECYP1A2
SCHEMBL18865595 0.68 HRH4 (0.47) ALDH1A1HRH3KDM4EHRH4
SCHEMBL16247101 0.67 ADORA2A (0.34) ALDH1A1KDM4ECYP1A2MAPK1HSD17B10
SCHEMBL16410174 0.67 PLD1 (0.46) PLD1HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115996929-A Antagonists of adenosine A2a receptors 阿道尔克斯治疗有限公司 2023-04-21 CN disclosed