SCHEMBL28994342

SCHEMBL28994342

CC(C)(C)OC(=O)C1(c2cc(CN3CC(C(C(F)(F)F)C(F)(F)F)CC34CCN(C(=O)O)CC4)cc(C(F)(F)F)c2)CCCC1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 6/20 0.38
TACR1 P25103 2/20 0.37
CYP2D6 P10635 2/20 0.34
TSHR P16473 2/20 0.34
USP2 O75604 5/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2C19 P33261 2/20 0.34
ALDH1A1 P00352 2/20 0.34
CYP3A4 P08684 2/20 0.33
HPGD P15428 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28994340 0.81 MGLL (0.40) MGLLTACR1CYP2D6TSHRUSP2
SCHEMBL20769556 0.77 MGLL (0.61) MGLL
SCHEMBL29532670 0.77 MGLL (0.61) MGLL
SCHEMBL2374489 0.77 TACR1 (0.47) TACR1CYP2D6TSHRUSP2CYP1A2
SCHEMBL20769632 0.74 MGLL (0.43) MGLL
SCHEMBL28994325 0.74 MGLL (0.43) MGLLCYP2D6
SCHEMBL19975519 0.73 CYP2D6 (0.51) MGLLTACR1CYP2D6TSHRUSP2
SCHEMBL28304786 0.72 CYP3A4 (0.47) TACR1CYP2D6TSHRUSP2CYP1A2
SCHEMBL19974348 0.71 STS (0.30)
SCHEMBL28304841 0.70 CYP2D6 (0.42) MGLLTACR1CYP2D6TSHRUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111032034-B Spiro compounds and methods of making and using the same H.隆德贝克有限公司 2023-05-02 CN disclosed