SCHEMBL28996170

SCHEMBL28996170

Nc1ccnc(-c2nccs2)c1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.58
ASIC3 Q9UHC3 2/20 0.48
SYK P43405 7/20 0.44
SRC P12931 4/20 0.44
ZAP70 P43403 3/20 0.44
PDPK1 O15530 1/20 0.42
RAB9A P51151 1/20 0.42
LOXL2 Q9Y4K0 1/20 0.42
ALDH1A1 P00352 1/20 0.41
TSHR P16473 1/20 0.41
NOS1 P29475 1/20 0.41
HSD17B10 Q99714 1/20 0.41
ADORA2A P29274 2/20 0.40
ADORA1 P30542 1/20 0.40
CDK2 P24941 1/20 0.38
SPHK2 Q9NRA0 1/20 0.38
SPHK1 Q9NYA1 1/20 0.38
CYP2A6 P11509 1/20 0.38
SMPD3 Q9NY59 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29290789 0.85 HSP90AA1 (0.55) HSP90AA1ASIC3SYKSRCZAP70
SCHEMBL30252529 0.80 HSP90AA1 (0.56) HSP90AA1SYKSRCZAP70PDPK1
SCHEMBL30511083 0.79
SCHEMBL16440627 0.77 SPR (0.49) HSP90AA1SYKSRCZAP70PDPK1
SCHEMBL15668705 0.77 SYK (0.49) HSP90AA1SYKSRCZAP70PDPK1
SCHEMBL20911090 0.77 HSP90AA1 (0.49) HSP90AA1SYKSRCZAP70PDPK1
SCHEMBL314105 0.76 ASIC3 (0.67) HSP90AA1ASIC3RAB9AALDH1A1TSHR
SCHEMBL5705089 0.74 HSP90AA1 (0.46) HSP90AA1PDPK1RAB9ALOXL2ALDH1A1
SCHEMBL27986436 0.74 KDM5C (0.57) HSP90AA1SYK
SCHEMBL9132675 0.74 ASIC3 (0.64) HSP90AA1ASIC3RAB9AALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109843879-B Benzothiazole derivatives as DYRK1 inhibitors 药物治疗股份有限公司 2023-05-02 CN disclosed
CN-109651358-B 4-aminopyridine derivative, pharmaceutical composition, preparation method and application thereof 上海迪诺医药科技有限公司 2023-04-07 CN disclosed