SCHEMBL29002452

SCHEMBL29002452

c1ccc2c(-c3cn[nH]c3)cccc2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 1/20 0.52
AKT2 P31751 1/20 0.52
PDK2 Q15119 1/20 0.46
AURKA O14965 1/20 0.45
AURKB Q96GD4 1/20 0.45
INCENP Q9NQS7 1/20 0.45
TPX2 Q9ULW0 1/20 0.45
MCL1 Q07820 1/20 0.44
ROCK2 O75116 1/20 0.44
ROCK1 Q13464 1/20 0.44
TNF P01375 1/20 0.43
PIK3CA P42336 1/20 0.43
PIK3CB P42338 1/20 0.43
ILK Q13418 1/20 0.42
CLK2 P49760 3/20 0.42
HIPK1 Q86Z02 3/20 0.42
HIPK2 Q9H2X6 3/20 0.42
HIPK3 Q9H422 3/20 0.42
CLK4 Q9HAZ1 3/20 0.42
DYRK2 Q92630 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29276383 0.84 AKT1 (0.47) AKT1AKT2PDK2AURKAAURKB
SCHEMBL28546134 0.77 AKT1 (0.43) AKT1AKT2PDK2AURKAAURKB
SCHEMBL30823568 0.76 AKT2 (0.59) AKT1AKT2PDK2AURKAAURKB
SCHEMBL28552255 0.76 AKT2 (0.72) AKT1AKT2PDK2AURKAAURKB
SCHEMBL30823569 0.76 AKT2 (0.59) AKT1AKT2PDK2AURKAAURKB
SCHEMBL10901163 0.76 MCL1 (0.50) MCL1TNFKDM4EGSK3BCA12
SCHEMBL15507900 0.76 AURKA (0.41) AKT1AKT2PDK2AURKAAURKB
SCHEMBL22861262 0.75 MCL1 (0.52) AKT1AKT2MCL1ROCK2ROCK1
SCHEMBL30144924 0.75 METAP2 (0.67) AKT1AKT2AURKAAURKBINCENP
SCHEMBL38660231 0.75 PRKCZ (0.59) AKT1AKT2AURKBROCK2CLK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116139936-A Carbonic anhydrase artificial enzyme and preparation method and application thereof 四川大学 2023-05-23 CN claimed
CN-116139936-B Carbonic anhydrase artificial enzyme and preparation method and application thereof 四川大学 2023-07-04 CN disclosed
CN-116139936-B Carbonic anhydrase artificial enzyme and preparation method and application thereof 四川大学 2023-07-04 CN disclosed
CN-116139936-A Carbonic anhydrase artificial enzyme and preparation method and application thereof 四川大学 2023-05-23 CN disclosed
CN-116139936-A Carbonic anhydrase artificial enzyme and preparation method and application thereof 四川大学 2023-05-23 CN disclosed