SCHEMBL29006256

SCHEMBL29006256

Cn1nccc1C(C(=O)NC(F)(F)F)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OXTR P30559 1/20 0.41
AVPR1A P37288 1/20 0.41
TACR1 P25103 2/20 0.36
PDE2A O00408 1/20 0.35
CYP3A4 P08684 4/20 0.35
NPSR1 Q6W5P4 1/20 0.35
KLRK1 P26718 1/20 0.35
MICA Q29983 1/20 0.35
RAET1L Q5VY80 1/20 0.35
LDHA P00338 1/20 0.35
LDHB P07195 1/20 0.35
CES2 O00748 1/20 0.35
CES1 P23141 1/20 0.35
CNR2 P34972 1/20 0.34
CYP26A1 O43174 1/20 0.34
SMO Q99835 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29006282 0.89 HDAC3 (0.41)
SCHEMBL29006269 0.86 OXTR (0.41) OXTRAVPR1ATACR1PDE2ACYP3A4
SCHEMBL29006259 0.86 NPSR1 (0.44) TACR1CYP3A4NPSR1KLRK1MICA
SCHEMBL29006260 0.85 CNR1 (0.39) NPSR1CNR2
SCHEMBL29006257 0.80 HDAC4 (0.46) NPSR1CES2CES1CNR2CYP26A1
SCHEMBL29006270 0.79 CNR2 (0.39) NPSR1CNR2SMO
SCHEMBL29006264 0.77 TDP1 (0.40) CYP3A4NPSR1MEN1KMT2A
SCHEMBL29006280 0.77 HDAC4 (0.41) MEN1KMT2A
SCHEMBL29006265 0.75 HTT (0.38) NPSR1MEN1KMT2A
SCHEMBL29006258 0.71 HDAC3 (0.42) NPSR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116003323-B Fluorine-containing pyrazole phenylacetamide derivative and application thereof 西北农林科技大学 2023-12-08 CN disclosed
CN-116003323-A Fluorine-containing pyrazole phenylacetamide derivative and application thereof 西北农林科技大学 2023-04-25 CN disclosed