SCHEMBL29006264

SCHEMBL29006264

COc1cccc(C(C(=O)NC(F)(F)F)c2ccnn2C)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GPR139 Q6DWJ6 2/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ROCK2 O75116 6/20 0.38
ROCK1 Q13464 6/20 0.38
PRKG1 Q13976 3/20 0.38
CHEK1 O14757 2/20 0.38
RPS6KA5 O75582 2/20 0.38
PRKCG P05129 2/20 0.38
CDK1 P06493 2/20 0.38
PRKACA P17612 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29006260 0.86 CNR1 (0.39) ALDH1A1LMNAHTTSMN1; SMN2NPSR1
SCHEMBL29006279 0.86 ALDH1A1 (0.43) TDP1ALDH1A1GPR139MTNR1AMTNR1B
SCHEMBL29006257 0.85 HDAC4 (0.46) MEN1POLBKMT2ANPSR1RPS6KB1
SCHEMBL29006259 0.84 NPSR1 (0.44) ALDH1A1MEN1LMNAPOLBKMT2A
SCHEMBL29006265 0.79 HTT (0.38) TDP1ALDH1A1MEN1POLBHTT
SCHEMBL29006282 0.78 HDAC3 (0.41) TDP1LMNAPOLBSMN1; SMN2MAPK1
SCHEMBL29006256 0.77 OXTR (0.41) MEN1KMT2ANPSR1CYP3A4
SCHEMBL17865258 0.75 PKM (0.54) MTNR1AMTNR1B
SCHEMBL29006270 0.74 CNR2 (0.39) LMNAPOLBNPSR1MAPK1
SCHEMBL29006280 0.74 HDAC4 (0.41) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116003323-B Fluorine-containing pyrazole phenylacetamide derivative and application thereof 西北农林科技大学 2023-12-08 CN disclosed
CN-116003323-A Fluorine-containing pyrazole phenylacetamide derivative and application thereof 西北农林科技大学 2023-04-25 CN disclosed