SCHEMBL29008490

SCHEMBL29008490

CCCc1c[nH]c(-c2cccc(C(F)(F)F)c2)n1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 4/20 0.57
CTSS P25774 2/20 0.57
PIN1 Q13526 1/20 0.47
HRH1 P35367 1/20 0.47
HRH4 Q9H3N8 1/20 0.47
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 1/20 0.45
SCN2A Q99250 1/20 0.45
CXCR2 P25025 1/20 0.44
TLR8 Q9NR97 1/20 0.44
GRK6 P43250 1/20 0.44
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
THRB P10828 1/20 0.43
PKM P14618 1/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3012997 0.86 HRH1 (0.60) CTSKCTSSPIN1HRH1HRH4
SCHEMBL31093434 0.86 CTSK (0.52) CTSKCTSSPIN1HRH1HRH4
SCHEMBL3023938 0.86 CTSK (0.52) CTSKCTSSPIN1HRH1HRH4
SCHEMBL535052 0.78 PDE5A (0.44) CTSKPIN1KDM4ENPC1ALDH1A1
SCHEMBL27642887 0.77 SCN2A (0.51) CTSSPIN1HRH1HRH4CYP1A2
SCHEMBL4446189 0.76 CTSK (0.67) CTSKCTSSTLR8XDHKCNH2
SCHEMBL7667716 0.75 MEN1 (0.55) PIN1CYP1A2GRK6KDM4EMEN1
SCHEMBL26467068 0.73 IDO1 (0.49) CTSKCTSSPIN1HRH1HRH4
SCHEMBL31659840 0.73 IDO1 (0.49) CTSKCTSSPIN1HRH1HRH4
SCHEMBL7192429 0.73 KIF11 (0.44) CTSKCTSSPIN1CXCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116194537-A Combination therapy with adenosine receptor antagonists 泰昂治疗公司 2023-05-30 CN disclosed