SCHEMBL29010909

SCHEMBL29010909

CC(C)c1ccc(COc2cccc(C3NC(=O)c4ccccc4N3)c2)cc1

nearest known ligand 0.78

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TNKS2 Q9H2K2 11/20 0.78
TNKS O95271 2/20 0.61
PARP3 Q9Y6F1 2/20 0.61
EGFR P00533 1/20 0.60
MAPT P10636 2/20 0.52
GAA P10253 1/20 0.52
ALDH1A1 P00352 2/20 0.46
KDM4E B2RXH2 1/20 0.46
HPGD P15428 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
MAPK1 P28482 1/20 0.43
AR P10275 1/20 0.41
MAOA P21397 1/20 0.41
ACHE P22303 1/20 0.41
MAOB P27338 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29010782 0.88 EGFR (0.77) TNKS2TNKSPARP3EGFRMAPT
SCHEMBL29010891 0.88 TNKS2 (0.83) TNKS2EGFRMAPTGAAALDH1A1
SCHEMBL29010778 0.88 TNKS2 (0.83) TNKS2EGFRMAPTGAAALDH1A1
SCHEMBL29010903 0.88 TNKS2 (1.00) TNKS2EGFRMAPTGAAALDH1A1
SCHEMBL29010896 0.86 TNKS2 (0.83) TNKS2EGFRMAPTGAAALDH1A1
SCHEMBL29010775 0.86 TNKS2 (0.83) TNKS2EGFRMAPTGAAALDH1A1
SCHEMBL29010780 0.79 TNKS2 (0.76) TNKS2TNKSPARP3EGFRMAPT
SCHEMBL27925475 0.76 TNKS2 (0.72) TNKS2TNKSPARP3MAPTGAA
SCHEMBL2821455 0.76 TNKS2 (0.72) TNKS2TNKSPARP3MAPTGAA
SCHEMBL27925494 0.76 TNKS2 (0.72) TNKS2TNKSPARP3MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116178283-B 2-Phenyl-2, 3-dihydro-quinazolin-4 (1H) -one derivative, preparation and application thereof 武汉科技大学 2024-07-02 CN disclosed
CN-116178283-A 2-phenyl-2, 3-dihydro-quinazolin-4 (1H) -one derivative, preparation and application thereof 武汉科技大学 2023-05-30 CN disclosed