SCHEMBL29010780

SCHEMBL29010780

CC(C)c1ccc(COc2ccccc2C2NC(=O)c3ccccc3N2)cc1

nearest known ligand 0.76

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TNKS2 Q9H2K2 13/20 0.76
TNKS O95271 1/20 0.58
PARP3 Q9Y6F1 1/20 0.58
EGFR P00533 1/20 0.52
ALDH1A1 P00352 4/20 0.49
KDM4E B2RXH2 3/20 0.49
HPGD P15428 3/20 0.49
HSD17B10 Q99714 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
TSHR P16473 1/20 0.49
PBRM1 Q86U86 1/20 0.49
KMT2A Q03164 3/20 0.43
CYP1A2 P05177 1/20 0.43
NPC1 O15118 1/20 0.43
MAPT P10636 1/20 0.41
MEN1 O00255 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29010900 0.87 TNKS2 (0.81) TNKS2EGFRALDH1A1KDM4EHPGD
SCHEMBL29010899 0.87 TNKS2 (0.81) TNKS2EGFRALDH1A1KDM4EHPGD
SCHEMBL29010889 0.87 TNKS2 (1.00) TNKS2EGFRALDH1A1KDM4EHPGD
SCHEMBL29010888 0.86 TNKS2 (0.83) TNKS2EGFRALDH1A1KDM4EHPGD
SCHEMBL29010776 0.85 TNKS2 (0.81) TNKS2EGFRALDH1A1KDM4EHPGD
SCHEMBL29010782 0.82 EGFR (0.77) TNKS2TNKSPARP3EGFRALDH1A1
SCHEMBL29010909 0.79 TNKS2 (0.78) TNKS2TNKSPARP3EGFRALDH1A1
SCHEMBL15033492 0.76 TNKS2 (0.60) TNKS2TNKSPARP3ALDH1A1KDM4E
SCHEMBL7670240 0.75 TNKS2 (0.65) TNKS2TNKSPARP3ALDH1A1KDM4E
SCHEMBL3770937 0.73 RXRA (0.54) KDM4EMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116178283-B 2-Phenyl-2, 3-dihydro-quinazolin-4 (1H) -one derivative, preparation and application thereof 武汉科技大学 2024-07-02 CN disclosed
CN-116178283-A 2-phenyl-2, 3-dihydro-quinazolin-4 (1H) -one derivative, preparation and application thereof 武汉科技大学 2023-05-30 CN disclosed