SCHEMBL290110

SCHEMBL290110

CS(=O)(=O)c1cccc(-c2ccc(C(C#N)CNC(=O)C3(NC(=O)O)CCOCC3)cc2)c1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSC P53634 5/20 0.56
CTSL P07711 13/20 0.46
CTSS P25774 12/20 0.46
CTSK P43235 12/20 0.46
CTSB P07858 10/20 0.46
CTSF Q9UBX1 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL290312 0.86 CTSC (0.41) CTSCCTSLCTSSCTSKCTSB
SCHEMBL289590 0.85 CTSC (0.38) CTSCCTSLCTSSCTSKCTSB
SCHEMBL2890791 0.84 CTSC (0.77) CTSCCTSLCTSSCTSKCTSB
SCHEMBL290266 0.83 CTSC (0.38) CTSCCTSLCTSSCTSKCTSB
SCHEMBL290666 0.82 CTSC (0.38) CTSCCTSLCTSSCTSKCTSB
SCHEMBL290024 0.82 CTSC (0.49) CTSCCTSLCTSSCTSKCTSB
SCHEMBL288986 0.82 MMP1 (0.41) CTSCCTSLCTSSCTSKCTSB
SCHEMBL290246 0.81 ALDH1A1 (0.41) CTSCCTSLCTSSCTSKCTSB
SCHEMBL290432 0.81 CTSL (0.46) CTSLCTSSCTSB
SCHEMBL290579 0.80 CTSL (0.47) CTSCCTSLCTSSCTSKCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP disclosed
WO-2010128324-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 ASTRAZENECA AB (SE) 2010-11-11 WO disclosed