SCHEMBL29011983

SCHEMBL29011983

CCOc1ccncc1Oc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 4/20 0.54
PTGS2 P35354 3/20 0.54
LTA4H P09960 1/20 0.50
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
TSPO P30536 4/20 0.44
ALB P02768 1/20 0.44
AOC3 Q16853 2/20 0.42
OPRK1 P41145 2/20 0.41
GLA P06280 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29011979 0.84 L3MBTL1 (0.51) PTGS1PTGS2CA12CA1CA2
SCHEMBL3819637 0.82 CA12 (0.58) CA12CA1CA2CA9CA14
SCHEMBL17077468 0.80 LMNA (0.49)
SCHEMBL11738087 0.80 LTA4H (0.63) LTA4HGLAL3MBTL1
SCHEMBL9488090 0.77 PTGS1 (0.51) PTGS1PTGS2TSPOALBOPRK1
SCHEMBL9339338 0.75 PTGS1 (0.58) PTGS1PTGS2LTA4HTSPOOPRK1
SCHEMBL21105143 0.75 PTGS1 (0.50) PTGS1PTGS2LTA4HTSPOOPRK1
SCHEMBL1078323 0.73 LTA4H (0.50) LTA4HGLAL3MBTL1
SCHEMBL17101823 0.73 GRM5 (0.43)
SCHEMBL2506700 0.73 CYP1A2 (0.52) PTGS1PTGS2TSPOL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111527078-B Pyridinecarbonyl derivatives and their therapeutic use as TRPC6 inhibitors 勃林格殷格翰国际公司 2023-06-02 CN disclosed