SCHEMBL29016575

SCHEMBL29016575

FC(F)Oc1ccc(Cc2nc3ccc(N=C(c4ccccc4)c4ccccc4)cc3s2)cc1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 1/20 0.34
HTT P42858 1/20 0.34
PDE10A Q9Y233 1/20 0.34
KMT2A Q03164 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
GRM2 Q14416 1/20 0.34
PPARG P37231 4/20 0.33
PPARA Q07869 4/20 0.33
MAPT P10636 3/20 0.33
TP53 P04637 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP3A4 P08684 1/20 0.33
TSHR P16473 1/20 0.33
SCD O00767 1/20 0.32
LIPG Q9Y5X9 1/20 0.32
AKR1A1 P14550 1/20 0.32
AKR1B1 P15121 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29016639 0.86 CSNK1D (0.40) MRGPRX4KMT2AHDAC6MAPTTP53
SCHEMBL30370383 0.86 CSNK1D (0.40) MRGPRX4KMT2AHDAC6MAPTTP53
SCHEMBL29016646 0.81 PSEN1 (0.39) KMT2AMAPTSMN1; SMN2CYP3A4LIPG
SCHEMBL30370198 0.81 PSEN1 (0.39) KMT2AMAPTSMN1; SMN2CYP3A4LIPG
SCHEMBL29016628 0.79 KDM4E (0.47) MRGPRX4HTTKMT2AHDAC6PPARA
SCHEMBL30370793 0.79 KDM4E (0.47) MRGPRX4HTTKMT2AHDAC6PPARA
SCHEMBL29016638 0.77 GPR52 (0.43) MAPTSMN1; SMN2LIPGAKR1B1
SCHEMBL29016559 0.76 MAPT (0.43) KMT2AMAPTTP53SMN1; SMN2CYP3A4
SCHEMBL29016596 0.76 PPARA (0.40) HTTPDE10AKMT2AHDAC6PPARA
SCHEMBL30370454 0.76 PPARA (0.40) HTTPDE10AKMT2AHDAC6PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108689942-B Nitrogen-containing bicyclic compound, and preparation method and application thereof 广东东阳光药业有限公司 2023-06-09 CN disclosed