SCHEMBL29016646

SCHEMBL29016646

N#Cc1ccc(Cc2nc3ccc(N=C(c4ccccc4)c4ccccc4)cc3s2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 1/20 0.39
PSEN2 P49810 1/20 0.39
APH1B Q8WW43 1/20 0.39
NCSTN Q92542 1/20 0.39
APH1A Q96BI3 1/20 0.39
PSENEN Q9NZ42 1/20 0.39
POLB P06746 1/20 0.39
CYP2C9 P11712 1/20 0.38
CYP3A4 P08684 1/20 0.38
ALDH1A1 P00352 1/20 0.37
CYP2C19 P33261 1/20 0.37
LIPG Q9Y5X9 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
APP P05067 2/20 0.35
LCK P06239 1/20 0.35
ITK Q08881 1/20 0.35
AURKB Q96GD4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30370198 1.00 PSEN1 (0.39) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL29016575 0.81 MRGPRX4 (0.34) CYP3A4LIPGSMN1; SMN2MAPTKMT2A
SCHEMBL29016639 0.81 CSNK1D (0.40) CYP2C9CYP3A4SMN1; SMN2MAPTKMT2A
SCHEMBL30370383 0.81 CSNK1D (0.40) CYP2C9CYP3A4SMN1; SMN2MAPTKMT2A
SCHEMBL29016548 0.78 KDM4E (0.50) POLBCYP2C9CYP3A4ALDH1A1CYP2C19
SCHEMBL30370795 0.78 KDM4E (0.50) POLBCYP2C9CYP3A4ALDH1A1CYP2C19
SCHEMBL29016638 0.77 GPR52 (0.43) ALDH1A1LIPGSMN1; SMN2MAPTNPC1
SCHEMBL30370212 0.74 APP (0.54) POLBCYP2C9CYP3A4ALDH1A1CYP2C19
SCHEMBL29016610 0.74 APP (0.54) POLBCYP2C9CYP3A4ALDH1A1CYP2C19
SCHEMBL30370846 0.74 CYP2C9 (0.45) POLBCYP2C9CYP3A4ALDH1A1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108689942-B Nitrogen-containing bicyclic compound, and preparation method and application thereof 广东东阳光药业有限公司 2023-06-09 CN disclosed