SCHEMBL2902355

SCHEMBL2902355

COc1ccc(-c2nc3ccccc3n2Cc2c(C)cccc2C)c(OCC(N)=O)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 5/20 0.44
KDM4E B2RXH2 5/20 0.44
LMNA P02545 4/20 0.44
NPSR1 Q6W5P4 2/20 0.44
CTSD P07339 2/20 0.44
MAPT P10636 5/20 0.43
TP53 P04637 5/20 0.43
TSHR P16473 3/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
ALDH1A1 P00352 4/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
CNR2 P34972 1/20 0.43
HPGD P15428 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
PLA2G2A P14555 2/20 0.41
MMP2 P08253 1/20 0.40
GAA P10253 1/20 0.40
PKM P14618 1/20 0.40
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2901560 0.90 NPSR1 (0.42) HTTKDM4ELMNANPSR1MAPT
SCHEMBL2907639 0.88 PLA2G2A (0.44) HTTKDM4ELMNANPSR1CTSD
SCHEMBL639847 0.87 KDM4E (0.50) HTTKDM4ELMNANPSR1MAPT
SCHEMBL2905631 0.83 LMNA (0.51) HTTKDM4ELMNANPSR1CTSD
SCHEMBL2905371 0.83 POLB (0.46) HTTKDM4ELMNANPSR1TP53
SCHEMBL2910004 0.81 ALDH1A1 (0.45) HTTKDM4ELMNANPSR1MAPT
SCHEMBL2906933 0.81 NPSR1 (0.53) HTTKDM4ELMNANPSR1MAPT
SCHEMBL638972 0.79 BRD4 (0.41) HTTKDM4ELMNANPSR1MEN1
SCHEMBL2901531 0.79 PLA2G2A (0.44) HTTKDM4ELMNANPSR1MAPT
SCHEMBL2903474 0.78 KMT2A (0.42) HTTKDM4ELMNANPSR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121627-B1 BENZIMIDAZOLE DERIVATIVES MERCK PATENT GMBH (DE) 2010-08-18 EP claimed
EP-2121627-A1 BENZIMIDAZOLE DERIVATIVES Merck Patent GmbH (DE) 2009-11-25 EP claimed
WO-2008101586-A1 BENZIMIDAZOLE DERIVATIVES MERCK PATENT GMBH (DE) 2008-08-28 WO claimed