SCHEMBL29025136

SCHEMBL29025136

Cn1cc(-c2ncnc(Cl)n2)c2ccccc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.47
POLB P06746 1/20 0.47
CTDSP1 Q9GZU7 1/20 0.47
CDK2 P24941 2/20 0.47
CCNE2 O96020 1/20 0.47
CDK4 P11802 1/20 0.47
CCND1 P24385 1/20 0.47
CCNE1 P24864 1/20 0.47
ALDH1A1 P00352 2/20 0.46
PRKCA P17252 1/20 0.46
GSK3B P49841 1/20 0.46
ABCB1 P08183 1/20 0.46
ABCG2 Q9UNQ0 1/20 0.46
CCNT1 O60563 2/20 0.46
CDK9 P50750 2/20 0.46
CDK5 Q00535 2/20 0.45
CDK5R1 Q15078 2/20 0.45
NPC1 O15118 1/20 0.45
LMNA P02545 1/20 0.45
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3362091 0.84 KDM4E (0.63) KDM4EPOLBCTDSP1CDK2CCNE2
SCHEMBL22509195 0.83 GSK3B (0.44) KDM4EPOLBCDK2CDK4CCND1
SCHEMBL30705248 0.83 GSK3B (0.44) KDM4EPOLBCDK2CDK4CCND1
SCHEMBL24240371 0.82 GSK3B (0.34) KDM4ECDK2GSK3BABCB1ABCG2
SCHEMBL22509160 0.82 GSK3B (0.46) KDM4EPOLBCDK2ALDH1A1PRKCA
SCHEMBL30705246 0.82 GSK3B (0.46) KDM4EPOLBCDK2ALDH1A1PRKCA
SCHEMBL29212194 0.79 BRD4 (0.48) KDM4ECDK2CCNE2CDK4CCND1
SCHEMBL5096322 0.79 MKNK1 (0.50) KDM4ECDK2ALDH1A1CCNT1CDK9
SCHEMBL29419125 0.79 MKNK1 (0.50) KDM4ECDK2ALDH1A1CCNT1CDK9
SCHEMBL22509188 0.79 GSK3B (0.49) KDM4EALDH1A1PRKCAGSK3BCDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110357863-B Triazine double aromatic ring derivative epidermal growth factor inhibitor and preparation method and application thereof 药雅科技(上海)有限公司 2023-04-14 CN disclosed