SCHEMBL29029059

SCHEMBL29029059

COc1ccc(CNS(=O)(=O)c2ccc(N(C)OS(C)(=O)=O)c([N+](=O)[O-])c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
CYP19A1 P11511 2/20 0.47
TSHR P16473 2/20 0.47
LMNA P02545 2/20 0.47
HTT P42858 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
USP2 O75604 1/20 0.46
ALDH3A1 P30838 1/20 0.46
VCAM1 P19320 1/20 0.46
CNR2 P34972 1/20 0.45
POLB P06746 1/20 0.44
MCOLN3 Q8TDD5 1/20 0.44
KDM4E B2RXH2 1/20 0.44
MAPK1 P28482 1/20 0.44
THRB P10828 1/20 0.42
RECQL P46063 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29471221 0.84 ALDH1A1 (0.47) ALDH1A1CYP19A1TSHRLMNAHTT
SCHEMBL29029080 0.83 ALDH1A1 (0.49) ALDH1A1CYP19A1TSHRLMNAHTT
SCHEMBL29029071 0.83 ALDH1A1 (0.49) ALDH1A1CYP19A1TSHRLMNAHTT
SCHEMBL29029090 0.81 TSHR (0.49) ALDH1A1CYP19A1TSHRLMNAHTT
SCHEMBL26547989 0.79 KDM4E (0.60) ALDH1A1CYP19A1TSHRLMNAHTT
SCHEMBL30480910 0.78 ALDH3A1 (0.60) ALDH1A1CYP19A1TSHRLMNAHTT
SCHEMBL4911967 0.74 ALDH1A1 (0.70) ALDH1A1CYP19A1TSHRLMNAHTT
SCHEMBL28156680 0.74 MEN1 (0.71) ALDH1A1CYP19A1TSHRPOLBRECQL
SCHEMBL11637929 0.73 NPC1 (0.59) ALDH1A1CYP19A1TSHRLMNAHTT
SCHEMBL15660010 0.73 MAPT (0.54) ALDH1A1CYP19A1TSHRLMNACNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116368128-A Heterocyclic compounds as CBP/EP300 bromodomain inhibitors 奥瑞基尼肿瘤有限公司 2023-06-30 CN disclosed