SCHEMBL2902927

SCHEMBL2902927

CC(C)N1CCN(CCCCN2CCN(C(=O)/C=C/c3ccc(F)c(Cl)c3)CCC2=O)CC1C

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PYGL P06737 3/20 0.42
GPR183 P32249 5/20 0.41
ITGB2 P05107 2/20 0.39
ICAM1 P05362 2/20 0.39
ITGAL P20701 2/20 0.39
CCR2 P41597 2/20 0.38
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2902206 0.93 GPR183 (0.47) PYGLGPR183CCR2
SCHEMBL2904553 0.91 GPR183 (0.47) PYGLGPR183CCR2
SCHEMBL2905175 0.87 PYGL (0.47) PYGLGPR183ITGB2ICAM1ITGAL
SCHEMBL2899437 0.84 CCR2 (0.42) PYGLGPR183ITGB2ICAM1ITGAL
SCHEMBL2904597 0.84 CCR2 (0.44) PYGLGPR183ITGB2ICAM1ITGAL
SCHEMBL2898977 0.83 PYGL (0.42) PYGLGPR183ITGB2ICAM1ITGAL
SCHEMBL2898974 0.83 PYGL (0.42) PYGLGPR183ITGB2ICAM1ITGAL
SCHEMBL2898971 0.83 PYGL (0.42) PYGLGPR183ITGB2ICAM1ITGAL
SCHEMBL2899701 0.83 CCR2 (0.42) PYGLGPR183ITGB2ICAM1ITGAL
SCHEMBL2898969 0.83 PYGL (0.42) PYGLGPR183ITGB2ICAM1ITGAL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010506-B1 DIAZEPAN DERIVATIVES MODULATORS OF CHEMOKINE RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-04 EP disclosed