SCHEMBL290305

SCHEMBL290305

Cc1c(Cl)ncnc1OC1CCCCN1C(=O)OC(C)C

nearest known ligand 0.45

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 20/20 0.45
CYP2C9 P11712 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL288924 0.85 GPR119 (0.33) GPR119
SCHEMBL288948 0.81 GPR119 (0.65) GPR119CYP2C9
SCHEMBL1445594 0.80 GPR119 (0.40) GPR119CYP2C9
SCHEMBL6066337 0.80 GPR119 (0.58) GPR119CYP2C9
SCHEMBL10120902 0.76 GPR119 (0.67) GPR119
SCHEMBL10106329 0.76 GPR119 (0.67) GPR119
SCHEMBL12277411 0.73 GPR119 (0.67) GPR119CYP2C9
SCHEMBL12277466 0.73 GPR119 (0.67) GPR119CYP2C9
SCHEMBL12236456 0.73 GPR119 (0.69) GPR119CYP2C9
SCHEMBL6456096 0.73 GPR119 (0.54) GPR119CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2504342-A1 IMIDAZO-PYRAZOLES AS GPR119 INHIBITORS Pfizer Inc. (US) 2012-10-03 EP disclosed
EP-2480551-A1 GPR 119 MODULATORS Pfizer Inc. (US) 2012-08-01 EP disclosed
EP-2427448-A1 Gpr 119 modulators Pfizer Inc. (US) 2012-03-14 EP disclosed
WO-2011061679-A1 IMIDAZO-PYRAZOLES AS GPR119 INHIBITORS PFIZER INC. (US) 2011-05-26 WO disclosed
WO-2011036576-A1 GPR 119 MODULATORS PFIZER INC. (US) 2011-03-31 WO disclosed
WO-2010128414-A1 GPR 119 MODULATORS PFIZER INC. (US) 2010-11-11 WO disclosed