SCHEMBL29033979

SCHEMBL29033979

Fc1[c]ccc(-c2ccc(Cl)c(Cl)c2)c1Cl

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 6/20 0.53
CYP1B1 Q16678 1/20 0.44
PSEN1 P49768 2/20 0.37
PSEN2 P49810 2/20 0.37
APH1B Q8WW43 2/20 0.37
NCSTN Q92542 2/20 0.37
APH1A Q96BI3 2/20 0.37
PSENEN Q9NZ42 2/20 0.37
APP P05067 2/20 0.37
DHFR P00374 1/20 0.36
AKR1C3 P42330 3/20 0.35
AKR1C2 P52895 3/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
SCN9A Q15858 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
NOTUM Q6P988 2/20 0.33
PTGER1 P34995 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5967116 0.83 AHR (0.59) AHRCYP1B1PSEN1PSEN2APH1B
SCHEMBL15225447 0.79 AHR (0.47) AHRCYP1B1PSEN1PSEN2APH1B
SCHEMBL7821465 0.76 CYP2A6 (0.40)
SCHEMBL20134691 0.74 PTGS2 (0.45) NPC1RAB9AMEN1KMT2A
SCHEMBL17515013 0.71 NISCH (0.38) NPC1RAB9AKDM4EMEN1GAA
SCHEMBL17514936 0.71 ABL1 (0.41) CYP1B1AKR1C3AKR1C2CYP3A4CYP2C9
SCHEMBL2282125 0.70 AHR (1.00) AHRCYP1B1PSEN1PSEN2APH1B
SCHEMBL224657 0.69
SCHEMBL22463151 0.69 AHR (0.46) AHRCYP1B1PSEN1PSEN2APH1B
SCHEMBL17514538 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116234546-A GPX4 inhibitors, pharmaceutical compositions thereof and their use in the treatment of GPX4 mediated diseases 嘉兴优博生物技术有限公司 2023-06-06 CN claimed