SCHEMBL29034858

SCHEMBL29034858

Cc1ccc2c(c1)c1c(n2-c2ccc(C(F)(F)F)cc2)CCC(C(=O)O)C1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.51
AKR1C2 P52895 3/20 0.51
AKR1C4 P17516 1/20 0.43
PTGS1 P23219 1/20 0.43
AKR1C1 Q04828 1/20 0.43
NOTUM Q6P988 1/20 0.41
HTR6 P50406 2/20 0.41
HRH1 P35367 1/20 0.41
PTGDR2 Q9Y5Y4 8/20 0.40
TEAD1 P28347 1/20 0.38
TEAD4 Q15561 1/20 0.38
TEAD2 Q15562 1/20 0.38
TEAD3 Q99594 1/20 0.38
HSD17B10 Q99714 2/20 0.37
USP2 O75604 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
ALOX15 P16050 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30500624 1.00 AKR1C3 (0.51) AKR1C3AKR1C2AKR1C4PTGS1AKR1C1
SCHEMBL11836738 0.75 AKR1C3 (0.67) AKR1C3AKR1C2AKR1C4PTGS1AKR1C1
SCHEMBL11837225 0.74 AKR1C3 (0.63) AKR1C3AKR1C2AKR1C4PTGS1AKR1C1
SCHEMBL11834560 0.74 AKR1C3 (0.72) AKR1C3AKR1C2AKR1C4PTGS1AKR1C1
SCHEMBL11837722 0.74 AKR1C3 (0.62) AKR1C3AKR1C2AKR1C4PTGS1AKR1C1
SCHEMBL13368695 0.74 HTR6 (0.67) HTR6HRH1
SCHEMBL30500623 0.73 HTR6 (0.47) HTR6HRH1PTGDR2TEAD1
SCHEMBL29034622 0.73 HTR6 (0.47) HTR6HRH1PTGDR2TEAD1
SCHEMBL30500622 0.73 HTR6 (0.49) HTR6HRH1ALDH1A1
SCHEMBL13011561 0.73 PTGDR2 (0.52) AKR1C3AKR1C2AKR1C4PTGS1AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116425670-A Novel heterocyclic compounds as TEAD inhibitors 英矽智能科技(上海)有限公司 2023-07-14 CN disclosed