SCHEMBL290368

SCHEMBL290368

CC(C)(C)OC(=O)NC1(C(=O)N(N)[C@H](C=O)Cc2ccc(I)cc2)CCOCC1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 1/20 0.35
ATM Q13315 1/20 0.31
RET P07949 1/20 0.31
CTSC P53634 1/20 0.30
KCNH2 Q12809 1/20 0.30
LTB4R Q15722 1/20 0.30
LTB4R2 Q9NPC1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL290586 0.85 CTSC (0.34) CTSCKCNH2LTB4RLTB4R2
SCHEMBL2893107 0.78 TACR2 (0.40)
SCHEMBL2893105 0.78 TACR2 (0.40)
SCHEMBL2890517 0.76 CTSC (0.48) RETCTSCKCNH2LTB4RLTB4R2
SCHEMBL2890519 0.76 CTSC (0.48) RETCTSCKCNH2LTB4RLTB4R2
SCHEMBL290369 0.75 GHSR (0.32) GHSRRET
SCHEMBL16485828 0.68 GRB2 (0.40)
SCHEMBL16478335 0.68 GRB2 (0.40)
SCHEMBL16478334 0.68 GRB2 (0.40)
SCHEMBL7223168 0.68 KLK5 (0.45) ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP disclosed
WO-2010128324-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 ASTRAZENECA AB (SE) 2010-11-11 WO disclosed