SCHEMBL29040796

SCHEMBL29040796

N#Cc1ccc2c(c1)CCCN(C(=O)O)C2

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 2/20 0.50
AKR1C1 Q04828 1/20 0.50
NAMPT P43490 9/20 0.46
DRD2 P14416 2/20 0.45
DRD3 P35462 2/20 0.45
HDAC6 Q9UBN7 4/20 0.43
USP30 Q70CQ3 2/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29040828 0.94 AKR1C3 (0.50) AKR1C3AKR1C1NAMPTDRD2DRD3
SCHEMBL29040775 0.91 AKR1C3 (0.52) AKR1C3AKR1C1NAMPTDRD2DRD3
SCHEMBL28369820 0.85 AKR1C3 (0.52) AKR1C3AKR1C1NAMPTDRD2DRD3
SCHEMBL566589 0.85 NAMPT (0.54) AKR1C3AKR1C1NAMPTUSP30
SCHEMBL20720388 0.82 AKR1C3 (0.48) AKR1C3AKR1C1NAMPTDRD2DRD3
SCHEMBL2995065 0.81 ESR2 (0.59) AKR1C3AKR1C1NAMPTDRD2DRD3
SCHEMBL17797626 0.78 BRD4 (0.49) NAMPTHDAC6HDAC8
SCHEMBL1263462 0.78 ABHD6 (0.50) AKR1C3NAMPTHDAC6HDAC8
SCHEMBL21762279 0.76 DRD2 (0.56) AKR1C3AKR1C1DRD2DRD3
SCHEMBL24265587 0.76 NR1H2 (0.58) AKR1C3NAMPTDRD2DRD3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116507326-A Compounds as GLP-1R agonists 拓臻制药公司 2023-07-28 CN disclosed